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第 42 卷第 3 期Vol. 42 No. 3
2012 年 6 月Jun 2012

所屬欄目:專(zhuān)論與綜述

N-苯基甘氨酸酯衍生物的合成與生物活性研究進(jìn)展
陳前進(jìn),王培義,李艷飛,冉義江,吳志兵* (綠色農藥與生物工程國家重點(diǎn)實(shí)驗室培育基地和教育部重點(diǎn)實(shí)驗室,貴州大學(xué) 精細化工研究開(kāi)發(fā)中心,貴州 貴陽(yáng)550025)
摘 要:綜述了近10年來(lái)具有良好生物活性的N-苯基甘氨酸酯衍生物的國內外研究進(jìn)展,簡(jiǎn)單討論其結構與生物活性(農藥活性和醫藥活性之間)的關(guān)系,并對其發(fā)展趨勢和應用前景作了展望。
關(guān)鍵詞:N-苯基甘氨酸酯;生物活性;研究進(jìn)展
中圖分類(lèi)號:S482.2+6  文獻標識碼:A  文章編號:1009-9212(2012)03-0001-05
Research Progress on Synthesis and Bioactivity of N-Phenyl Glycine Ester Derivatives
CHEN Qian-jin,WANG Pei-yi,LI Yan-fei,Ran Yi-jiang,Wu Zhi-bing* (Key Laboratory of Green Pesticide and Agricultural Bioengineering,Ministry of Education;Center for Research and Development of Fine Chemicals,Guizhou University,Guiyang 550025,China)
Abstract:The research progresses on synthesis and bioactivities of N-phenyl glycine ester derivatives were reviewed. The discussion was organized into two parts based on medicinal and agrochemical bioactivities. The structure and activity relationship of the title compounds were discussed briefly. The development tendency as well as the prospect of N-phenyl glycine ester derivatives was summarized.
Key words:N-Phenyl glycine ester;biological activity;research progress
作者簡(jiǎn)介:陳前進(jìn)(1981-),男,貴州德江人,碩士研究生,研究方向:有機合成。(E-mail:362283891@qq.com)
聯(lián) 系 人:吳志兵,講師,研究方向:農藥創(chuàng )制。(E-mail:wzb1171@163.com)
收稿日期:2012-03-31
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